{"id":1929,"date":"2019-12-22T16:48:59","date_gmt":"2019-12-22T15:48:59","guid":{"rendered":"https:\/\/www.ayrmed.com\/editorial\/?p=1929"},"modified":"2019-12-22T16:49:07","modified_gmt":"2019-12-22T15:49:07","slug":"ecdisteroides-evidencias-cientificas","status":"publish","type":"post","link":"https:\/\/www.ayrmed.com\/editorial\/ecdisteroides-evidencias-cientificas\/","title":{"rendered":"Ecdisteroides. Evidencias cient\u00edficas"},"content":{"rendered":"<p style=\"text-align: justify;\">Al echar un vistazo a la composici\u00f3n de ciertos preparados de gran \u00e9xito en tiendas nutricionales, vemos a menudo que su propaganda carece de toda base cient\u00edfica, pues se anuncian supuestas propiedades en relaci\u00f3n con la presencia de compuestos sobre los que en realidad a\u00fan no se ha demostrado cient\u00edficamente ning\u00fan beneficio objetivo en humanos. Tal es el caso de los ecdisteroides y su presunto papel como \u00abanabolizantes naturales\u00bb.<\/p>\n<p style=\"text-align: center;\"><a href=\"https:\/\/www.ayrmed.com\/editorial\/wp-content\/uploads\/2019\/12\/ecdisteroides.png\"><img loading=\"lazy\" decoding=\"async\" class=\"alignnone size-full wp-image-1930\" src=\"https:\/\/www.ayrmed.com\/editorial\/wp-content\/uploads\/2019\/12\/ecdisteroides.png\" alt=\"ecdisteroides\" width=\"496\" height=\"325\" srcset=\"https:\/\/www.ayrmed.com\/editorial\/wp-content\/uploads\/2019\/12\/ecdisteroides.png 496w, https:\/\/www.ayrmed.com\/editorial\/wp-content\/uploads\/2019\/12\/ecdisteroides-300x197.png 300w\" sizes=\"auto, (max-width: 496px) 100vw, 496px\" \/><\/a><\/p>\n<p style=\"text-align: center;\"><!--more--><\/p>\n<p style=\"text-align: justify;\">Los ecdisteroides ejercen varios efectos farmacol\u00f3gicos beneficiosos en los mam\u00edferos. Seg\u00fan la literatura cient\u00edfica, su capacidad para aumentar la s\u00edntesis proteica parece ser el m\u00e1s prominente, y es comparable a la de los esteroides anabolico-androg\u00e9nicos. Adem\u00e1s, los ecdisteroides poseen otros beneficios importantes, tales como:<\/p>\n<ul style=\"text-align: justify;\">\n<li>Baja toxicidad para vertebrados. El consumo inofensivo de verduras con alto contenido en ecdisteroides (como la espinaca, la quinoa o la casta\u00f1a), y de los preparados que contienen ecdiesteroides, es prueba de su seguridad.<\/li>\n<li>Estas mol\u00e9culas\u00a0no se unen a los receptores de esteroides nucleares de vertebrados (estrog\u00e9nicos, glucocorticoides y andr\u00f3genos), lo que significa que no ejercen efectos secundarios hormonales caracter\u00edsticos de los esteroides anab\u00f3licos androg\u00e9nicos. Estos datos\u00a0relevantes tambi\u00e9n fueron apoyados por los resultados de los ensayos de uni\u00f3n de radioligando.<\/li>\n<li>Los par\u00e1metros farmacocin\u00e9ticos de los ecdisteroides son favorables, debido a su alta polaridad y relativamente alta hidrosolubilidad. Esta propiedad es fundamental en los procedimientos de dise\u00f1o famacol\u00f3gicos modernos.<\/li>\n<\/ul>\n<p>No obstante, a\u00fan quedan por resolverse algunas dudas importantes con respecto a esto compuestos:<\/p>\n<ul style=\"text-align: justify;\">\n<li>El mecanismo de acci\u00f3n es casi completamente desconocido.<\/li>\n<li>La cifra\u00a0de ecdisteroides conocidos est\u00e1 cerca de 300, lo que representa una gran variabilidad estructural. Dado que el perfil de la actividad depende bastante\u00a0de la estructura, se necesitan muchos m\u00e1s estudios para establecer una relaci\u00f3n estructura-actividad adecuada para determinar su verdadero papel como anabolizante\u00a0y la aparici\u00f3n de posibles efectos secundarios.<\/li>\n<li>Hay pocos\u00a0estudios disponibles en humanos, todos ellos con muy pocos pacientes en\u00a0periodos\u00a0de corta duraci\u00f3n, y en idioma ruso. A pesar de ello, cientos de preparados y\u00a0productos anab\u00f3licos que contienen ecdisteroides se anuncian comercialmente en Internet. Su dudoso origen, la legislaci\u00f3n y la composici\u00f3n de estos productos no los convierte en relevantes para sacar conclusiones sobre la eficacia y la seguridad terap\u00e9utica de los ecdisteroides en humanos.<\/li>\n<\/ul>\n<h2 style=\"text-align: center;\">Conclusiones sobre la utilidad de los ecdisteroides<\/h2>\n<p style=\"text-align: justify;\">En resumen, con la aclaraci\u00f3n de los aspectos mencionados anteriormente, algunos ecdisteroides podr\u00edan\u00a0convertirse en un futuro en alternativas terap\u00e9uticas prometedoras frente a\u00a0los esteroides anab\u00f3lico-androg\u00e9nicos. El uso prospectivo de ecdisteroides podr\u00eda\u00a0extenderse a tratamientos de condiciones patol\u00f3gicas en las que habitualmente se aplican los esteroides anab\u00f3licos, como por ejemplo para neutralizar el efecto de los glucocorticoides en las miopat\u00edas. Este tipo de aplicaciones valiosas pueden dar m\u00e1s importancia y actualidad a la investigaci\u00f3n en ecdisteroides.<\/p>\n<p style=\"text-align: justify;\">Asumir como\u00a0ciertas determinadas informaciones que pululan en p\u00e1ginas no confiables de Internet, en ciertos gimnasios y en algunas tiendas nutricionales puede convertir al consumidor en una verdadera cobaya o conejillo de indias, a menos que se esfuerce en buscar fuentes de informaci\u00f3n seguras y de aceptable\u00a0calidad cient\u00edfica.<\/p>\n<p style=\"text-align: center;\">\n<p style=\"text-align: justify;\">Fuente bibliogr\u00e1fica: <a href=\"http:\/\/www.eurekaselect.com\/66157\/article\" target=\"_blank\" rel=\"noopener noreferrer\">B\u00e1thori M,\u00a0T\u00f3th N,\u00a0Hunyadi A,\u00a0M\u00e1rki A,\u00a0Z\u00e1dor E. Phytoecdysteroids\u00a0and\u00a0anabolic-androgenic\u00a0steroids&#8211;structure\u00a0and\u00a0effects\u00a0on\u00a0humans. Curr Med Chem.\u00a02008;15(1):75-91.<\/a><\/p>\n","protected":false},"excerpt":{"rendered":"<p>Al echar un vistazo a la composici\u00f3n de ciertos preparados de gran \u00e9xito en tiendas nutricionales, vemos a menudo que su propaganda carece de toda base cient\u00edfica, pues se anuncian supuestas propiedades en relaci\u00f3n con la presencia de compuestos sobre los que en realidad a\u00fan no se ha demostrado cient\u00edficamente ning\u00fan beneficio objetivo en humanos. [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"site-sidebar-layout":"default","site-content-layout":"","ast-site-content-layout":"default","site-content-style":"default","site-sidebar-style":"default","ast-global-header-display":"","ast-banner-title-visibility":"","ast-main-header-display":"","ast-hfb-above-header-display":"","ast-hfb-below-header-display":"","ast-hfb-mobile-header-display":"","site-post-title":"","ast-breadcrumbs-content":"","ast-featured-img":"","footer-sml-layout":"","ast-disable-related-posts":"","theme-transparent-header-meta":"","adv-header-id-meta":"","stick-header-meta":"","header-above-stick-meta":"","header-main-stick-meta":"","header-below-stick-meta":"","astra-migrate-meta-layouts":"default","ast-page-background-enabled":"default","ast-page-background-meta":{"desktop":{"background-color":"","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-opacity":"","overlay-gradient":""},"tablet":{"background-color":"","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-opacity":"","overlay-gradient":""},"mobile":{"background-color":"","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-opacity":"","overlay-gradient":""}},"ast-content-background-meta":{"desktop":{"background-color":"var(--ast-global-color-5)","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-opacity":"","overlay-gradient":""},"tablet":{"background-color":"var(--ast-global-color-5)","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-opacity":"","overlay-gradient":""},"mobile":{"background-color":"var(--ast-global-color-5)","background-image":"","background-repeat":"repeat","background-position":"center center","background-size":"auto","background-attachment":"scroll","background-type":"","background-media":"","overlay-type":"","overlay-color":"","overlay-opacity":"","overlay-gradient":""}},"footnotes":""},"categories":[2],"tags":[],"class_list":["post-1929","post","type-post","status-publish","format-standard","hentry","category-dietas-personalizadas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.4 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Ecdisteroides, \u00bffuncionan realmente? | Ayrmed.com<\/title>\n<meta name=\"description\" content=\"Ecdisteroides y fitoecdisteroides. 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